SCHEMBL8557068

SCHEMBL8557068

Cc1ccccc1NC(=O)Nc1ccc(C(=O)N2Cc3ccccc3Cc3ccccc32)cc1

nearest known ligand 0.72

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 3/20 0.57
AVPR1A P37288 3/20 0.57
MAPT P10636 2/20 0.52
RAB9A P51151 2/20 0.52
NPC1 O15118 1/20 0.52
MEN1 O00255 1/20 0.49
HTT P42858 1/20 0.49
KMT2A Q03164 1/20 0.49
OXTR P30559 1/20 0.48
NAMPT P43490 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562633 0.88 AVPR2 (0.55) AVPR2AVPR1ARAB9ANPC1HTT
SCHEMBL8560800 0.83 AVPR2 (0.79) AVPR2AVPR1AOXTR
SCHEMBL7363716 0.83 AVPR1A (0.66) AVPR2AVPR1A
SCHEMBL7344881 0.82 AVPR1A (0.72) AVPR2AVPR1AOXTR
SCHEMBL8556275 0.81 AVPR2 (0.69) AVPR2AVPR1AOXTR
SCHEMBL8563072 0.80 SMN1; SMN2 (0.55) AVPR2AVPR1AMAPTRAB9ANPC1
SCHEMBL8560873 0.79 ACHE (0.60) AVPR2AVPR1ARAB9ANAMPT
SCHEMBL9236961 0.79 AVPR2 (0.66) AVPR2AVPR1AOXTR
SCHEMBL8558733 0.78 AVPR2 (0.65) AVPR2AVPR1AOXTR
SCHEMBL8564119 0.78 AVPR2 (0.68) AVPR2AVPR1AMEN1KMT2AOXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed