SCHEMBL8563072

SCHEMBL8563072

Cc1cccc(NC(=O)c2ccc(C(=O)N3Cc4ccccc4Cc4ccccc43)cc2)c1C

nearest known ligand 0.66

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.55
AVPR2 P30518 2/20 0.52
AVPR1A P37288 2/20 0.52
NAMPT P43490 1/20 0.48
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
MAPT P10636 3/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
LMNA P02545 1/20 0.47
THRB P10828 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562633 0.92 AVPR2 (0.55) SMN1; SMN2AVPR2AVPR1ANPC1RAB9A
SCHEMBL8562828 0.84 AVPR2 (0.49) SMN1; SMN2AVPR2AVPR1ANPC1RAB9A
SCHEMBL8562097 0.84 AVPR2 (0.49) SMN1; SMN2AVPR2AVPR1ANPC1RAB9A
SCHEMBL8557607 0.83 NPC1 (0.50) AVPR2AVPR1ANPC1RAB9AMAPT
SCHEMBL8556275 0.83 AVPR2 (0.69) AVPR2AVPR1A
SCHEMBL8558857 0.83 HPGD (0.57) SMN1; SMN2NAMPTNPC1RAB9AMEN1
SCHEMBL7333170 0.83 AVPR1A (0.66) AVPR2AVPR1A
SCHEMBL8557068 0.80 AVPR2 (0.57) AVPR2AVPR1ANAMPTNPC1RAB9A
SCHEMBL8560873 0.79 ACHE (0.60) AVPR2AVPR1ANAMPTRAB9A
SCHEMBL8560800 0.79 AVPR2 (0.79) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed