SCHEMBL8555842

SCHEMBL8555842

O=C1[N]c2cc(F)ccc2NC1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.39
LRRK2 Q5S007 3/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA12 O43570 1/20 0.38
CA4 P22748 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
TGM2 P21980 2/20 0.36
MEN1 O00255 1/20 0.36
FLT3 P36888 1/20 0.36
CCNE1 P24864 2/20 0.36
CDK2 P24941 2/20 0.36
CCNE2 O96020 1/20 0.36
CYP1A2 P05177 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C19 P33261 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
CHRM1 P11229 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6264592 0.81 CA1 (0.40) KMT2ALRRK2CA1CA2CA12
SCHEMBL4750469 0.81 CA1 (0.40) KMT2ALRRK2CA1CA2CA12
SCHEMBL2429783 0.79 JUN (0.44) KMT2A
SCHEMBL8555812 0.78 TGM2 (0.50) KMT2ALRRK2TGM2MEN1FLT3
SCHEMBL8556891 0.78 RET (0.37) KMT2ACA1CA2CA12CA9
SCHEMBL5760370 0.78 ROS1 (0.46) KMT2ALRRK2CA1CA2CA12
SCHEMBL8121964 0.77
SCHEMBL8558339 0.75 PDPK1 (0.45) LRRK2CCNB2CDK1CCNB1CCNB3
SCHEMBL8555149 0.74 CA1 (0.39) CA1CA2CA12CA9TGM2
SCHEMBL2334055 0.73 EPHX2 (0.41) TGM2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647137-A4 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF. UNIV CALIFORNIA WEBER ECKARD (US) 1998-09-16 EP disclosed
EP-0647137-A1 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-04-12 EP disclosed