SCHEMBL8557318

SCHEMBL8557318

CCc1cc[c]c(-c2ccc(C(=N)N)cc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 5/20 0.48
ALDH1A1 P00352 1/20 0.41
TOP1 P11387 1/20 0.41
HPGD P15428 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PRMT1 Q99873 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
TOP2A P11388 1/20 0.40
TOP2B Q02880 1/20 0.40
PRSS1 P07477 4/20 0.40
PRSS2 P07478 3/20 0.40
PRSS3 P35030 3/20 0.40
F10 P00742 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.40
WDR5 P61964 1/20 0.40
F2 P00734 1/20 0.37
PLG P00747 1/20 0.37
PLAU P00749 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8176603 0.85 NQO2 (0.48) NQO2ALDH1A1TOP1HPGDCASP1
SCHEMBL8088676 0.80 NOTUM (0.39) ALDH1A1
SCHEMBL5320671 0.77 HSD17B10 (0.33) ALDH1A1HPGDHSD17B10TDP1
SCHEMBL8169371 0.77 PLAU (0.38) NQO2PRSS1PRSS2PRSS3F10
SCHEMBL7191695 0.76 NQO2 (0.44) NQO2ALDH1A1TOP1HPGDCASP1
SCHEMBL8169396 0.76 NQO2 (0.44) NQO2ALDH1A1TOP1HPGDCASP1
SCHEMBL4463655 0.76 MAPT (0.32) ALDH1A1
SCHEMBL1371003 0.75 TP53 (0.43) ALDH1A1
SCHEMBL7154087 0.74 NPC1 (0.37)
SCHEMBL15067982 0.74 TRPA1 (0.39) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832076-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-04-01 EP disclosed