SCHEMBL8169396

SCHEMBL8169396

N=C(N)c1ccc(-c2[c]ccc(I)c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 4/20 0.44
ALDH1A1 P00352 1/20 0.44
TOP1 P11387 1/20 0.44
HPGD P15428 1/20 0.44
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PRMT1 Q99873 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
TOP2A P11388 1/20 0.43
TOP2B Q02880 1/20 0.43
WDR5 P61964 1/20 0.43
LMNA P02545 1/20 0.38
MASP2 O00187 1/20 0.38
PLAU P00749 1/20 0.38
THPO P40225 1/20 0.38
F2 P00734 1/20 0.37
PRSS1 P07477 1/20 0.37
APEX1 P27695 1/20 0.37
PRSS3 P35030 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7191695 0.80 NQO2 (0.44) NQO2ALDH1A1TOP1HPGDCASP1
SCHEMBL8557318 0.76 NQO2 (0.48) NQO2ALDH1A1TOP1HPGDCASP1
SCHEMBL8485694 0.74 WDR5 (0.57) NQO2ALDH1A1TOP1HPGDCASP1
SCHEMBL8169720 0.73 C1S (0.44) NQO2ALDH1A1TOP1HPGDCASP1
SCHEMBL8170510 0.73 NQO2 (0.44) NQO2ALDH1A1TOP1HPGDCASP1
SCHEMBL8174039 0.73 NQO2 (0.43) NQO2ALDH1A1TOP1HPGDCASP1
SCHEMBL8169108 0.73 LMNA (0.48) NQO2ALDH1A1TOP1HPGDCASP1
SCHEMBL11501514 0.73 ALDH1A1 (0.33) ALDH1A1
SCHEMBL10449127 0.73 ACHE (0.32) ALDH1A1HPGDHSD17B10TDP1LMNA
SCHEMBL6189586 0.72 ALDH1A1 (0.33) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114328-A ANTICOAGULANTS; BLOOD DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-09-05 US disclosed
US-5849736-A Isoxazoline and isoxazole fibrinogen receptor antagonists THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-12-15 US disclosed
EP-0730590-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-11 EP disclosed