SCHEMBL8557623

SCHEMBL8557623

O=C(O)NC1(CI)NCCc2ccccc21

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HCAR2 Q8TDS4 1/20 0.35
KIF11 P52732 3/20 0.33
EDNRB P24530 1/20 0.33
EDNRA P25101 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
OPRM1 P35372 1/20 0.33
TSHR P16473 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HTR2A P28223 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561279 0.86 KIF11 (0.37) MEN1HDAC9HCAR2KIF11EDNRB
SCHEMBL8560374 0.84 MEN1 (0.35) MEN1HDAC9HCAR2KIF11EDNRB
SCHEMBL8560551 0.82 MEN1 (0.37) MEN1HDAC9KIF11
SCHEMBL8555341 0.75 ALDH1A1 (0.39) MEN1HDAC9HCAR2KIF11EDNRB
SCHEMBL27852609 0.69 ALDH1A1 (0.41) MEN1HDAC9HCAR2TSHRNPSR1
SCHEMBL28312964 0.68 TDP1 (0.40) MEN1HDAC9HCAR2TSHRNPSR1
SCHEMBL28008400 0.67 HDAC9 (0.41) MEN1HDAC9HCAR2KIF11TSHR
SCHEMBL27969858 0.67 MEN1 (0.40) MEN1HDAC9HCAR2TSHRNPSR1
SCHEMBL7201343 0.67 ALDH1A1 (0.39) MEN1HDAC9HCAR2KIF11TSHR
SCHEMBL9845298 0.67 ALDH1A1 (0.60) MEN1HDAC9HCAR2EDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0538248-B1 TETRAHYDROISOQUINOLINYLCARBAMATES OF 1,2,3,3A,8,8A-HEXAHYDRO-1,3A,8-TRIMETHYLPYRROLO [2,3-B]INDOLE HOECHST MARION ROUSSEL INC (US) 1998-02-11 EP claimed