SCHEMBL8557834

SCHEMBL8557834

NC(=O)CN1CCN(Cc2nc(-c3ccc(F)cc3)c(-c3ccc(F)cc3)o2)CC1c1c(Cl)cc(N)cc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC29A1 Q99808 1/20 0.36
SCN9A Q15858 1/20 0.36
GRM2 Q14416 3/20 0.34
NR4A2 P43354 1/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
GAA P10253 1/20 0.34
RXRA P19793 6/20 0.33
RXRB P28702 6/20 0.33
RXRG P48443 6/20 0.33
KCNK3 O14649 1/20 0.32
KCNK9 Q9NPC2 1/20 0.32
PTGS1 P23219 1/20 0.32
EPHX2 P34913 1/20 0.32
PTGS2 P35354 1/20 0.32
CNR1 P21554 1/20 0.32
CCR5 P51681 1/20 0.32
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553960 0.81 SLC29A1 (0.59) SLC29A1GAARXRARXRBRXRG
SCHEMBL8557836 0.78 SLC29A1 (0.43) SLC29A1GAAMEN1LMNAKMT2A
SCHEMBL8557838 0.78 KCNK3 (0.35) NR4A2RXRARXRBRXRGKCNK3
SCHEMBL8554772 0.73 SLC29A1 (0.53) SLC29A1NR4A2CYP3A4CYP2C19RXRA
SCHEMBL8552619 0.73 SLC29A1 (0.53) SLC29A1NR4A2CYP3A4CYP2C19RXRA
SCHEMBL8553498 0.69 SLC29A1 (0.49) SLC29A1NR4A2CYP3A4CYP2C19RXRA
SCHEMBL8553599 0.69 KDR (0.48) NR4A2CYP3A4CYP2C19GAARXRA
SCHEMBL8554766 0.66 KDR (0.45) SLC29A1NR4A2CYP3A4CYP2C19RXRA
SCHEMBL8598990 0.66 SLC29A1 (0.45) SLC29A1NR4A2CYP3A4CYP2C19RXRA
SCHEMBL18409631 0.65 KCNH2 (0.49) NR4A2CYP3A4CYP2C19RXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0582164-B1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles BRISTOL MYERS SQUIBB CO (US) 1998-12-23 EP claimed