SCHEMBL8557836

SCHEMBL8557836

Nc1cc(Cl)c(NC(=O)CN2CCN(Cc3nc(-c4ccc(F)cc4)c(-c4ccc(F)cc4)o3)CC2)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC29A1 Q99808 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
ALDH1A1 P00352 4/20 0.41
KMT2A Q03164 4/20 0.39
OGA O60502 1/20 0.39
KDR P35968 1/20 0.39
MEN1 O00255 2/20 0.39
TSHR P16473 2/20 0.39
USP2 O75604 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAP4K4 O95819 1/20 0.38
DRD4 P21917 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553599 0.91 KDR (0.48) NPC1RAB9AALDH1A1KMT2AKDR
SCHEMBL8553960 0.87 SLC29A1 (0.59) SLC29A1NPC1RAB9AALDH1A1KMT2A
SCHEMBL8557576 0.83 MEN1 (0.52) SLC29A1ALDH1A1KMT2AOGAMEN1
SCHEMBL8554568 0.81 KDR (0.58) ALDH1A1KMT2AKDRMEN1TSHR
SCHEMBL8557838 0.80 KCNK3 (0.35) ALDH1A1TSHRLMNAHTT
SCHEMBL8556969 0.79 REV1 (0.53) ALDH1A1KMT2AOGAKDRMEN1
SCHEMBL8554274 0.79 KDR (0.45) NPC1RAB9AALDH1A1KDRGAA
SCHEMBL8552619 0.79 SLC29A1 (0.53) SLC29A1KDRTSHRHPGDDRD4
SCHEMBL8553498 0.79 SLC29A1 (0.49) SLC29A1KDRTSHRHPGDDRD4
SCHEMBL8554772 0.79 SLC29A1 (0.53) SLC29A1KDRTSHRHPGDDRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0582164-B1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles BRISTOL MYERS SQUIBB CO (US) 1998-12-23 EP claimed
EP-0582164-A1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles Bristol-Myers Squibb Company (US) 1994-02-09 EP claimed