SCHEMBL8555748

SCHEMBL8555748

O=C1[N]c2cc([N+](=O)[O-])c(Br)cc2NC1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
MAPT P10636 3/20 0.40
XDH P47989 1/20 0.35
TYMS P04818 3/20 0.34
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
PKM P14618 1/20 0.33
CYP3A4 P08684 2/20 0.33
CAPN9 O14815 1/20 0.33
CASP3 P42574 1/20 0.33
MAPK1 P28482 1/20 0.32
CYP19A1 P11511 1/20 0.32
GLA P06280 1/20 0.32
GRIN2D O15399 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8128055 0.87 CYP3A4 (0.39) ALDH1A1MAPTGABRA1GABRG2GABRB3
SCHEMBL8118374 0.82 ESPL1 (0.38) ALDH1A1MAPTCYP3A4CAPN9CASP3
SCHEMBL8559761 0.82 AKR1B1 (0.40) ALDH1A1PKMCYP3A4CAPN9CASP3
SCHEMBL8554584 0.80 CES1 (0.38) BCHECES1
SCHEMBL8115079 0.79 ESPL1 (0.38) ALDH1A1MAPTCYP3A4CAPN9CASP3
SCHEMBL3672889 0.79 MAPT (0.37) ALDH1A1MAPTPKMCYP3A4CAPN9
SCHEMBL3670516 0.78 CA12 (0.40) ALDH1A1MAPTCYP3A4MAPK1GLA
SCHEMBL3675781 0.75 MAPT (0.48) ALDH1A1MAPTGRIN2DGRIN3BCYP1A2
SCHEMBL3678226 0.75 PTPN11 (0.44) MAPTCAPN9CASP3CYP1A2GRIA1
SCHEMBL8557868 0.74 CES1 (0.34) ALDH1A1MAPTTYMSBLMBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647137-A4 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF. UNIV CALIFORNIA WEBER ECKARD (US) 1998-09-16 EP disclosed
EP-0647137-A1 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-04-12 EP disclosed