SCHEMBL8558167

SCHEMBL8558167

CC(C)(C)OC(=O)NC(C(=O)Nc1ccccc1C(N)=O)c1ccc2c(c1)C(C)(C)CCC2(C)C

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
CYP26A1 O43174 1/20 0.39
CYP3A4 P08684 1/20 0.39
RARB P10826 1/20 0.39
RARG P13631 1/20 0.39
BACE1 P56817 3/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
PKM P14618 2/20 0.38
KDM4E B2RXH2 3/20 0.37
CTSL P07711 1/20 0.37
LMNA P02545 1/20 0.36
RXRA P19793 2/20 0.36
RXRB P28702 1/20 0.36
ALDH1A1 P00352 1/20 0.36
AAK1 Q2M2I8 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8102431 0.83 RARB (0.43) CTSSCTSKCYP26A1CYP3A4RARB
SCHEMBL8560537 0.80 CTSK (0.44) CTSSCTSKCYP26A1CYP3A4RARB
SCHEMBL8106743 0.79 MEN1 (0.42) CTSSCTSKCYP26A1CYP3A4RARB
SCHEMBL8757257 0.79 RARB (0.40) CTSSCTSKCYP26A1CYP3A4RARB
SCHEMBL8748829 0.78 RARB (0.55) CYP26A1CYP3A4RARBRARGMEN1
SCHEMBL8100983 0.78 RARB (0.44) CTSSCTSKCYP26A1CYP3A4RARB
SCHEMBL8555829 0.77 RARB (0.48) CYP26A1CYP3A4RARBRARGMEN1
SCHEMBL8100687 0.77 CYP3A4 (0.47) CYP3A4BACE1KMT2AALDH1A1
SCHEMBL8106311 0.77 RARB (0.37) CTSSCTSKCYP26A1CYP3A4RARB
SCHEMBL8561391 0.77 CTSS (0.48) CTSSCTSKCYP3A4RARGBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5709867-A TREATMENT OF DERMATOLOGICAL, RHEUMATIC, RESPIRATORY, CARDIOVASCULAR, AND OPHTHALMOLOGICAL DISORDERS CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 1998-01-20 US disclosed