SCHEMBL8558501

SCHEMBL8558501

CCCn1c2nc(CC)[nH]c2c(=O)n2nc(CC)nc12

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.45
ADORA2A P29274 2/20 0.44
ADORA2B P29275 2/20 0.44
SIRT1 Q96EB6 1/20 0.42
SIRT3 Q9NTG7 1/20 0.42
SIRT5 Q9NXA8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11389501 0.75 ADORA1 (0.61) ADORA1ADORA2AADORA2B
SCHEMBL8563310 0.75 ADORA2A (0.53) ADORA1ADORA2AADORA2B
SCHEMBL7951810 0.74 ADORA1 (0.53) ADORA1ADORA2AADORA2BSIRT1SIRT3
SCHEMBL8559082 0.71 ADORA1 (0.62) ADORA1ADORA2AADORA2B
SCHEMBL7414170 0.71 ADORA1 (0.52) ADORA1ADORA2AADORA2BSIRT1SIRT3
SCHEMBL4623457 0.71 ADORA2A (0.59) ADORA1ADORA2AADORA2BSIRT1SIRT3
SCHEMBL9430500 0.70 ADORA2A (0.60) ADORA1ADORA2AADORA2BSIRT1SIRT3
SCHEMBL7420292 0.69 ADORA1 (0.44) ADORA1ADORA2AADORA2BSIRT1SIRT3
SCHEMBL8560002 0.68 ADORA1 (0.58) ADORA1ADORA2AADORA2B
SCHEMBL27713795 0.68 SIRT1 (0.68) ADORA1ADORA2AADORA2BSIRT1SIRT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880524-A1 NEW TRIAZOLOPURINES, METHOD OF PREPARING THEM AND THEIR USE AS DRUGS Boehringer Ingelheim Pharma KG (DE) 1998-12-02 EP disclosed
WO-1998003511-A1 NEW TRIAZOLOPURINES, METHOD OF PREPARING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-01-29 WO disclosed