SCHEMBL8558960

SCHEMBL8558960

COc1cc2ncnc(Nc3ccc4nc(S(=O)(=O)Cc5ccccc5)[nH]c4c3)c2cc1OC

nearest known ligand 0.70

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 5/20 0.70
EGFR P00533 7/20 0.54
RET P07949 5/20 0.54
KDR P35968 3/20 0.54
LCK P06239 2/20 0.53
LRRK2 Q5S007 4/20 0.53
CLK1 P49759 1/20 0.52
ABCG2 Q9UNQ0 1/20 0.52
RIPK2 O43353 1/20 0.52
EPHB2 P29323 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558954 0.93 ERBB2 (0.63) ERBB2EGFRRETKDRLCK
SCHEMBL8093504 0.83 ERBB2 (0.70) ERBB2EGFRKDR
SCHEMBL8555757 0.83 ERBB2 (1.00) ERBB2EGFRRETKDRLCK
SCHEMBL8807988 0.82 EGFR (0.67) EGFRRETKDRLCKLRRK2
Hydrochloric Acid SCHEMBL8894722 0.82 ERBB2 (0.98) ERBB2EGFRRETKDRLCK
SCHEMBL8807285 0.80 EGFR (0.67) EGFRRETKDRLCKLRRK2
SCHEMBL8556343 0.80 KDR (0.72) ERBB2EGFRRETKDRLCK
Hydrochloric Acid SCHEMBL8896157 0.79 KDR (0.70) ERBB2EGFRRETKDRLCK
SCHEMBL5746250 0.76 AURKB (0.71) ERBB2EGFRKDR
SCHEMBL8555750 0.76 ERBB2 (0.87) ERBB2EGFRRETKDRLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP claimed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO claimed
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP disclosed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO disclosed