SCHEMBL8093504

SCHEMBL8093504

Nc1cc2c(Nc3ccc4nc(S(=O)(=O)Cc5ccccc5)[nH]c4c3)ncnc2cn1

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 4/20 0.70
EGFR P00533 3/20 0.47
KDR P35968 9/20 0.46
MET P08581 8/20 0.46
GRM1 Q13255 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558960 0.83 ERBB2 (0.70) ERBB2EGFRKDR
SCHEMBL8096012 0.81 ERBB2 (0.73) ERBB2EGFRKDRMETGRM1
SCHEMBL8558954 0.76 ERBB2 (0.63) ERBB2EGFRKDR
SCHEMBL8554234 0.75 MAPT (0.56)
SCHEMBL11965408 0.72 EGFR (0.78) ERBB2EGFRGRM1
SCHEMBL6765471 0.70 EGFR (0.53) ERBB2EGFR
SCHEMBL8554228 0.68 XDH (0.46)
SCHEMBL8082013 0.68 EGFR (0.74) ERBB2EGFRKDRGRM1
SCHEMBL8558474 0.68 ERBB2 (1.00) ERBB2EGFRKDRMET
SCHEMBL7209149 0.67 ALDH1A1 (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153617-A Irreversible bicyclic inhibitors of tyrosine kinases WARNER-LAMBERT COMPANY (US) 2000-11-28 US claimed
WO-1999006396-A1 IRREVERSIBLE BICYCLIC INHIBITORS OF TYROSINE KINASES WARNER-LAMBERT COMPANY (US) 1999-02-11 WO claimed
US-6153617-A Irreversible bicyclic inhibitors of tyrosine kinases WARNER-LAMBERT COMPANY (US) 2000-11-28 US disclosed
WO-1999006396-A1 IRREVERSIBLE BICYCLIC INHIBITORS OF TYROSINE KINASES WARNER-LAMBERT COMPANY (US) 1999-02-11 WO disclosed