SCHEMBL8559004

SCHEMBL8559004

COCCn1nc(-c2ccccc2)c2ccccc2c1=O

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.65
TSHR P16473 2/20 0.64
ALDH1A1 P00352 3/20 0.61
ALOX15 P16050 1/20 0.61
GAA P10253 2/20 0.57
TP53 P04637 2/20 0.57
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
MAPT P10636 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.56
POLB P06746 2/20 0.56
NPSR1 Q6W5P4 2/20 0.56
LMNA P02545 2/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
HTT P42858 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8864947 0.89 TP53 (0.71) RAB9AALDH1A1GAATP53MEN1
SCHEMBL8243795 0.81 ALDH1A1 (0.66) RAB9ATSHRALDH1A1ALOX15GAA
SCHEMBL3974796 0.80 SMN1; SMN2 (0.64) RAB9ATSHRALDH1A1ALOX15GAA
SCHEMBL13829609 0.79 ALDH1A1 (0.53) RAB9ATSHRALDH1A1GAATP53
SCHEMBL8555258 0.79 ALDH1A1 (0.73) RAB9ATSHRALDH1A1ALOX15GAA
SCHEMBL13729753 0.79 ALDH1A1 (0.53) RAB9ATSHRALDH1A1TP53MEN1
Hydrochloric Acid SCHEMBL4087801 0.79 SMN1; SMN2 (0.62) RAB9ATSHRALDH1A1ALOX15GAA
SCHEMBL7456859 0.77 PKM (0.52) RAB9ATSHRALDH1A1ALOX15GAA
SCHEMBL23755002 0.76 PTGS1 (0.45) RAB9ATSHRALDH1A1TP53MEN1
SCHEMBL7368621 0.76 ALDH1A1 (1.00) RAB9ATSHRALDH1A1ALOX15GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0475527-B1 Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents SANOFI SA (FR) 1998-02-25 EP disclosed
US-5624922-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1997-04-29 US disclosed
EP-0597540-B1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC (US) 1996-06-05 EP disclosed
US-5380721-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1995-01-10 US disclosed
EP-0597540-A1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1994-05-18 EP disclosed
EP-0475527-A2 Aryl-fused and hetaryl-fused-2, 4-diazepine and 2, 4-diazocine antiarrhythmic agents STERLING DRUG INC. (US) 1992-03-18 EP disclosed