SCHEMBL8559136

SCHEMBL8559136

CC(C)(C)OCC(O)CN1CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.57
ALDH1A1 P00352 4/20 0.57
TDP1 Q9NUW8 1/20 0.57
MAPT P10636 1/20 0.40
USP2 O75604 2/20 0.40
ALOX15 P16050 1/20 0.40
ABCB1 P08183 3/20 0.39
UGT8 Q16880 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
GLA P06280 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3970870 0.87 KDM4E (0.57) KDM4EALDH1A1TDP1MAPTUSP2
SCHEMBL3975409 0.87 KDM4E (0.57) KDM4EALDH1A1TDP1MAPTUSP2
SCHEMBL8559427 0.82 ALDH1A1 (0.49) KDM4EALDH1A1TDP1MAPTUSP2
SCHEMBL21667845 0.80 KDM4E (0.51) KDM4EALDH1A1TDP1MAPTL3MBTL1
SCHEMBL21667810 0.80 KMT2A (0.54) KDM4EALDH1A1TDP1MAPTL3MBTL1
SCHEMBL21667817 0.80 KDM4E (0.51) KDM4EALDH1A1TDP1MAPTL3MBTL1
SCHEMBL7277526 0.80 KMT2A (0.54) KDM4EALDH1A1TDP1MAPTL3MBTL1
SCHEMBL21743150 0.80 KDM4E (0.51) KDM4EALDH1A1TDP1MAPTL3MBTL1
SCHEMBL21667819 0.80 KMT2A (0.54) KDM4EALDH1A1TDP1MAPTL3MBTL1
SCHEMBL8745307 0.79 SMN1; SMN2 (0.58) KDM4EALDH1A1MAPTUSP2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700392-B1 USE OF MACROCYCLIC METAL COMPLEXES AS TEMPERATURE PROBES SCHERING AG (DE) 1998-12-09 EP disclosed
US-5747000-A 1,4-7-TRIS-(CARBOXYMETHYL)-1,4,7,10-TETRAAZACYCLODODECANE DERIVATIVES; DETERMINING CHEMICAL SHIFT OF SIGNALS IN NUCLEAR MAGNETIC RESONANCE SCHERING AKTIENGESELLSCHAFT (DE) 1998-05-05 US disclosed
EP-0596586-B1 Process for the production of metal complexes of N-beta-hydroxalkyl-tri-N-carboxyalkyl-1,4,7,10-tetraazacyclododecane and derivatives thereof SCHERING AG (DE) 1997-01-22 EP disclosed
EP-0700392-A1 USE OF MACROCYCLIC METAL COMPLEXES AS TEMPERATURE PROBES SCHERING AKTIENGESELLSCHAFT (DE) 1996-03-13 EP disclosed
US-5410043-A Chemical intermediate for metal complexes SCHERING AKTIENGESELLSCHAFT (DE) 1995-04-25 US disclosed
WO-1994027977-A1 USE OF MACROCYCLIC METAL COMPLEXES AS TEMPERATURE PROBES SCHERING AKTIENGESELLSCHAFT (DE) 1994-12-08 WO disclosed
EP-0596586-A1 Process for the production of metal complexes of N-beta-hydroxalkyl-tri-N-carboxyalkyl-1,4,7,10-tetraazacyclododecane and derivatives thereof SCHERING AKTIENGESELLSCHAFT (DE) 1994-05-11 EP disclosed