SCHEMBL8559646

SCHEMBL8559646

CS(=O)(=O)[N+]1(NC(=O)C(COCc2ccccc2)NC(=O)c2cccnc2)CC2(CCNCC2)c2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.38
LMNA P02545 2/20 0.36
ECE1 P42892 1/20 0.36
GPR132 Q9UNW8 6/20 0.35
BCL2 P10415 1/20 0.34
GHSR Q92847 1/20 0.34
CTSL P07711 2/20 0.34
CTSB P07858 2/20 0.34
CTSS P25774 2/20 0.34
RAB9A P51151 1/20 0.34
CTRC Q99895 1/20 0.34
CMKLR2 P46091 1/20 0.34
CMKLR1 Q99788 1/20 0.34
CTSK P43235 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561651 0.93 TACR1 (0.42) TACR1GHSR
SCHEMBL8560379 0.92 CTSL (0.40) TACR1GHSRCTSLCTSBCTSS
SCHEMBL8562715 0.89 TACR1 (0.41) TACR1
Hydrochloric Acid SCHEMBL8567968 0.88 TACR1 (0.41) TACR1
SCHEMBL8563536 0.88 TACR1 (0.45) TACR1GHSRCYP3A4
SCHEMBL8562851 0.87 TACR1 (0.43) TACR1CTSLCTSBCTSSCTSK
SCHEMBL8564711 0.87 TACR1 (0.43) TACR1GHSRCTSSCYP3A4
SCHEMBL8561512 0.87 CTSD (0.37) TACR1GHSRCTSS
SCHEMBL8559389 0.86 TACR1 (0.42) TACR1BCL2GHSRCTSLCTSS
Hydrochloric Acid SCHEMBL8560013 0.86 CTSD (0.37) TACR1GHSRCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811431-A Spiro-substituted azacyclic derivatives and their use as therapeutic agents MERCK SHARP & DOHME LTD. (GB) 1998-09-22 US disclosed