SCHEMBL8559684

SCHEMBL8559684

CCOC(=O)c1cn(C2CC2)c2c(C)c(N3CCN(C)CC3)c(F)c(Cl)c2c1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 1/20 0.43
ADRB2 P07550 1/20 0.43
ALDH1A1 P00352 3/20 0.41
HTT P42858 2/20 0.41
MAPK1 P28482 2/20 0.41
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
TSHR P16473 1/20 0.41
CASP1 P29466 1/20 0.41
KCNH2 Q12809 4/20 0.40
MAPK10 P53779 1/20 0.40
POLB P06746 2/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
WDR5 P61964 1/20 0.38
CACNA1F O60840 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8111823 0.92 STAT3 (0.45) STAT3ADRB2ALDH1A1HTTMAPK1
SCHEMBL8557811 0.88 MEN1 (0.51) ALDH1A1MAPK1MEN1KMT2AKCNH2
SCHEMBL8852491 0.83 STAT3 (0.44) STAT3ADRB2ALDH1A1HTTMAPK1
SCHEMBL9133982 0.83 ADRB2 (0.50) STAT3ADRB2ALDH1A1HTTMAPK1
SCHEMBL5704330 0.82 ADRB2 (0.49) STAT3ADRB2ALDH1A1HTTMAPK1
SCHEMBL8852028 0.82 STAT3 (0.43) STAT3ADRB2ALDH1A1HTTMAPK1
SCHEMBL10920186 0.82 ALDH1A1 (0.58) ADRB2ALDH1A1MAPK1MEN1KMT2A
SCHEMBL10572110 0.81 KCNH2 (0.60) ADRB2ALDH1A1MAPK1MEN1KMT2A
SCHEMBL8560598 0.81 ALDH1A1 (0.52) STAT3ADRB2ALDH1A1MAPK1LMNA
SCHEMBL7131518 0.80 ADRB2 (0.59) STAT3ADRB2ALDH1A1MAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0823413-A2 Benzoheterocyclic compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-02-11 EP disclosed
US-5591744-A 1,4-DIHYDRO-4-OXOQUINOLINE-3-CARBOXYLATE DERIVATIVES; MICROBIOCIDES OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1997-01-07 US disclosed
EP-0287951-B1 7-Piperazinyl- or 7-Morpholino-4-oxo-quinoline-3-carboxylic acid derivatives, their preparation and their use as antimicrobial agents OTSUKA PHARMA CO LTD (JP) 1996-07-03 EP disclosed
US-5495020-A CHEMICAL INTERMEDIATE FOR BACTERICIDES, MICROBIOCIDES, DISINFECTANTS; SIDE EFFECT REDUCTION, ABSORPTION OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1996-02-27 US disclosed
EP-0565132-A2 Benzoheterocyclic compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-10-13 EP disclosed
EP-0287951-A2 7-Piperazinyl- or 7-Morpholino-4-oxo-quinoline-3-carboxylic acid derivatives, their preparation and their use as antimicrobial agents OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1988-10-26 EP disclosed