SCHEMBL8560071

SCHEMBL8560071

CCCCN1CCC(c2sc3c(C(N)=O)c4ccccc4n3c2C)CC1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 1/20 0.41
CNR1 P21554 3/20 0.39
CNR2 P34972 3/20 0.39
HRH2 P25021 1/20 0.39
HTR7 P34969 5/20 0.39
PARP1 P09874 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PMP22 Q01453 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7449849 0.77 KDM4E (0.53) HTR4CNR1CNR2HTR7KDM4E
SCHEMBL8566824 0.69 HTR4 (0.47) HTR4HTR7KDM4EALDH1A1PMP22
SCHEMBL8521031 0.68 HTR4 (0.46) HTR4CNR1CNR2HTR7KDM4E
SCHEMBL8574546 0.68 HTR4 (0.46) HTR4HTR7KDM4EALDH1A1PMP22
SCHEMBL8575502 0.67 HTR4 (0.53) HTR4HRH2HTR7
SCHEMBL8520377 0.67 HTR4 (0.49) HTR4HRH2HTR7KDM4EALDH1A1
SCHEMBL1077431 0.66 HTR4 (0.50) HTR4HRH2HTR7
SCHEMBL7400351 0.65 HTR4 (0.43) HTR4HRH2KDM4EALDH1A1PMP22
SCHEMBL9345077 0.65 KDM4E (0.46) HTR4KDM4EALDH1A1PMP22NPSR1
SCHEMBL9342316 0.65 HTR4 (0.48) HTR4HTR7KDM4EALDH1A1PMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998409-A GASTROINTESTINAL DISORDERS; CARDIOVASCULAR DISORDERS; NERVOUS SYSTEM DISORDERS SMITHKLINE BEECHAM PLC (GB) 1999-12-07 US disclosed