SCHEMBL8574546

SCHEMBL8574546

CCCCN1CCC(C2(C)CCn3c(c(C(N)=O)c4ccccc43)S2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 2/20 0.46
HTR7 P34969 4/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
PMP22 Q01453 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CHRM1 P11229 2/20 0.37
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
HTR1A P08908 1/20 0.37
CHRM5 P08912 1/20 0.37
ADRA2A P08913 1/20 0.37
DRD2 P14416 1/20 0.37
ADRA2B P18089 1/20 0.37
CHRM3 P20309 1/20 0.37
DRD4 P21917 1/20 0.37
ADRA1D P25100 1/20 0.37
ADRA1A P35348 1/20 0.37
HRH1 P35367 1/20 0.37
ADRA1B P35368 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8566824 0.92 HTR4 (0.47) HTR4HTR7KDM4EALDH1A1PMP22
SCHEMBL8521031 0.82 HTR4 (0.46) HTR4HTR7KDM4EALDH1A1PMP22
SCHEMBL1077431 0.80 HTR4 (0.50) HTR4HTR7CHRM2ADRA2BHRH1
SCHEMBL8520377 0.77 HTR4 (0.49) HTR4HTR7KDM4EALDH1A1PMP22
SCHEMBL8575502 0.76 HTR4 (0.53) HTR4HTR7CHRM2ADRA2BHRH1
SCHEMBL8575712 0.76 HTR4 (0.47) HTR4HTR7CHRM2ADRA2BCHRM3
SCHEMBL7449849 0.71 KDM4E (0.53) HTR4HTR7KDM4EALDH1A1PMP22
SCHEMBL8574553 0.69 HTR2A (0.39) HTR4
SCHEMBL8560071 0.68 HTR4 (0.41) HTR4HTR7KDM4EALDH1A1PMP22
SCHEMBL7360838 0.68 HTR4 (0.49) HTR4KDM4EALDH1A1PMP22NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998409-A GASTROINTESTINAL DISORDERS; CARDIOVASCULAR DISORDERS; NERVOUS SYSTEM DISORDERS SMITHKLINE BEECHAM PLC (GB) 1999-12-07 US disclosed