Bromide

Bromide

SCHEMBL8560291

O=C1C([P+](c2ccccc2)(c2ccccc2)c2ccccc2)CCN1c1ccccc1F.[Br-]

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRM1 known ✓ P35372 2/20 0.35
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
FPR2 P25090 1/20 0.40
NOTUM Q6P988 1/20 0.39
KDM4E B2RXH2 1/20 0.37
ALOX15 P16050 1/20 0.37
KCNH2 Q12809 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
MGLL Q99685 1/20 0.35
GRM2 Q14416 1/20 0.33
LMNA P02545 1/20 0.33
HSD11B1 P28845 1/20 0.33
GRM5 P41594 1/20 0.33
OPRL1 P41146 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8898107 1.00 KMT2A (0.45) KMT2AMEN1FPR2NOTUMKDM4E
Bromide SCHEMBL8899375 0.89 NOTUM (0.35) KMT2AMEN1FPR2NOTUMKDM4E
Bromide SCHEMBL8567151 0.89 NOTUM (0.35) KMT2AMEN1FPR2NOTUMKDM4E
Bromide SCHEMBL8897674 0.81 ATM (0.51) KMT2AMEN1KDM4EOPRM1SIGMAR1
Bromide SCHEMBL8560897 0.81 ALDH1A1 (0.40) KMT2AMEN1KDM4ESIGMAR1LMNA
Bromide SCHEMBL8560903 0.81 ALDH1A1 (0.40) KMT2AMEN1KDM4ESIGMAR1LMNA
Bromide SCHEMBL8565603 0.81 ATM (0.51) KMT2AMEN1KDM4EOPRM1SIGMAR1
Bromide SCHEMBL7880298 0.81 MEN1 (0.43) KMT2AMEN1FPR2MGLL
Bromide SCHEMBL7880295 0.81 MEN1 (0.43) KMT2AMEN1FPR2MGLL
Bromide SCHEMBL8564801 0.79 ALDH1A1 (0.36) KMT2AKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0879237-A1 ISOOXACEPHEM DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1998-11-25 EP disclosed
US-5811419-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1998-09-22 US disclosed
US-5804577-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1998-09-08 US disclosed
WO-1997026260-A1 ISOOXACEPHEM DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-07-24 WO disclosed
EP-0761673-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed