SCHEMBL8560448

SCHEMBL8560448

CCOCc1nc(C(C)(C)O)c(C(=O)O)n1Cc1ccc(-c2ccccc2C(=O)C(=O)O)cc1

nearest known ligand 0.72

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 1/20 0.55
AGTR2 P50052 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7886323 0.94 AGTR1 (0.57) AGTR1AGTR2
SCHEMBL8566093 0.89 AGTR1 (0.68) AGTR1AGTR2
SCHEMBL8568722 0.87 AGTR1 (0.61) AGTR1AGTR2
SCHEMBL7878389 0.86 AGTR1 (0.52) AGTR1AGTR2
SCHEMBL7878411 0.86 AGTR1 (0.58) AGTR1AGTR2
Hydrochloric Acid SCHEMBL7887929 0.86 AGTR1 (0.51) AGTR1AGTR2
Hydrochloric Acid SCHEMBL8559318 0.85 AGTR1 (0.53) AGTR1AGTR2
SCHEMBL8561079 0.85 AGTR1 (0.49) AGTR1AGTR2
SCHEMBL7878738 0.85 AGTR1 (0.56) AGTR1AGTR2
SCHEMBL27348488 0.84 AGTR1 (0.54) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0603001-B1 Biphenyl derivatives, their preparation and their use for the treatment of hypertension and cardiac disease SANKYO CO (JP) 1998-08-26 EP disclosed
US-5459148-A Cardiovascular disorders SANKYO COMPANY, LIMITED (JP) 1995-10-17 US disclosed
EP-0603001-A1 Biphenyl derivatives, their preparation and their use for the treatment of hypertension and cardiac disease SANKYO COMPANY LIMITED (JP) 1994-06-22 EP disclosed