SCHEMBL8560936

SCHEMBL8560936

O=C1[C@@H](Br)CCN1c1cccnc1Cl

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.37
P2RX7 Q99572 3/20 0.36
ALDH1A1 P00352 4/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
TSHR P16473 1/20 0.35
ESR2 Q92731 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
LIPE Q05469 1/20 0.34
FPR1 P21462 1/20 0.34
FPR2 P25090 1/20 0.34
CYP2C19 P33261 1/20 0.33
MAPT P10636 1/20 0.33
FAAH O00519 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560932 1.00 GAA (0.37) GAAP2RX7ALDH1A1SMN1; SMN2TSHR
SCHEMBL28437828 0.78 HDAC1 (0.48) GAAALDH1A1MAPT
SCHEMBL8563081 0.76 KDM4E (0.39) ALDH1A1CYP2C19
SCHEMBL8563078 0.76 KDM4E (0.39) ALDH1A1CYP2C19
Bromide SCHEMBL8562114 0.75 GAA (0.35) GAAP2RX7ALDH1A1SMN1; SMN2TSHR
Bromide SCHEMBL8897946 0.75 GAA (0.35) GAAP2RX7ALDH1A1SMN1; SMN2TSHR
SCHEMBL7621523 0.74 CRBN (0.53) GAAALDH1A1SMN1; SMN2MAPTLMNA
SCHEMBL7621521 0.74 CRBN (0.53) GAAALDH1A1SMN1; SMN2MAPTLMNA
SCHEMBL7621516 0.74 CRBN (0.53) GAAALDH1A1SMN1; SMN2MAPTLMNA
SCHEMBL8560583 0.72 KMT2A (0.53) P2RX7ALDH1A1SMN1; SMN2TSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5804577-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1998-09-08 US disclosed
EP-0761673-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed