SCHEMBL8561603

SCHEMBL8561603

CN(CCCn1c(C=Cc2ccsc2)cc2ccccc21)C(=O)CC(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
CYP1A2 P05177 1/20 0.34
POLB P06746 1/20 0.34
HTR2A P28223 1/20 0.33
HTR2B P41595 1/20 0.33
NTRK1 P04629 1/20 0.33
CNR2 P34972 2/20 0.32
TSHR P16473 2/20 0.32
PPARA Q07869 1/20 0.32
HTT P42858 1/20 0.32
KDM4E B2RXH2 1/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TRPV4 Q9HBA0 2/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
HSP90AA1 P07900 1/20 0.31
MAPT P10636 1/20 0.31
GRK2 P25098 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561600 1.00 ALDH1A1 (0.34) ALDH1A1CYP1A2POLBHTR2AHTR2B
SCHEMBL8562540 0.77 HDAC1 (0.39) NTRK1CNR2TSHRMEN1NPC1
SCHEMBL8562543 0.77 HDAC1 (0.39) NTRK1CNR2TSHRMEN1NPC1
SCHEMBL8561161 0.74 MAPT (0.35) HTR2BNTRK1CNR2TSHRHTT
SCHEMBL8561158 0.74 MAPT (0.35) HTR2BNTRK1CNR2TSHRHTT
SCHEMBL10405577 0.69 ALDH1A1 (0.47) ALDH1A1CYP1A2POLBHTR2AHTR2B
SCHEMBL9832588 0.69 ALDH1A1 (0.47) ALDH1A1CYP1A2POLBHTR2AHTR2B
SCHEMBL8561604 0.69 PPARA (0.36) ALDH1A1TSHRPPARAKDM4ESMN1; SMN2
SCHEMBL8561601 0.69 PPARA (0.36) ALDH1A1TSHRPPARAKDM4ESMN1; SMN2
SCHEMBL5353392 0.60 ABCC2 (0.43) ALDH1A1CNR2HTTKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0695755-B1 Pyrrolocarbazole HOFFMANN LA ROCHE (CH) 1998-10-21 EP disclosed
EP-0695755-A1 Pyrrolocarbazoles F. Hoffmann-La Roche AG (CH) 1996-02-07 EP disclosed