SCHEMBL8562543

SCHEMBL8562543

OCCCn1c(C=Cc2ccsc2)cc2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.39
HDAC8 Q9BY41 3/20 0.39
CNR2 P34972 7/20 0.38
ALOX5 P09917 1/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
CNR1 P21554 1/20 0.35
NTRK1 P04629 1/20 0.33
NTRK3 Q16288 1/20 0.33
ABCC2 Q92887 1/20 0.32
NPC1 O15118 1/20 0.32
HSP90AA1 P07900 1/20 0.32
MAPT P10636 1/20 0.32
TSHR P16473 1/20 0.32
GRK2 P25098 1/20 0.32
RAB9A P51151 1/20 0.32
NR1H2 P55055 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562540 1.00 HDAC1 (0.39) HDAC1HDAC8CNR2ALOX5MEN1
SCHEMBL8561158 0.84 MAPT (0.35) CNR2ALOX5MEN1KMT2ANTRK1
SCHEMBL8561161 0.84 MAPT (0.35) CNR2ALOX5MEN1KMT2ANTRK1
SCHEMBL8561600 0.77 ALDH1A1 (0.34) CNR2MEN1KMT2ANTRK1NPC1
SCHEMBL8561603 0.77 ALDH1A1 (0.34) CNR2MEN1KMT2ANTRK1NPC1
SCHEMBL8561601 0.76 PPARA (0.36) NPC1MAPTTSHRRAB9A
SCHEMBL8561604 0.76 PPARA (0.36) NPC1MAPTTSHRRAB9A
SCHEMBL25145277 0.74 CNR2 (0.48) CNR2MEN1KMT2ACNR1ABCC2
SCHEMBL27366620 0.74 CNR2 (0.45) CNR2CNR1ABCC2TSHR
SCHEMBL9832588 0.68 ALDH1A1 (0.47) HDAC1HDAC8KMT2ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0695755-B1 Pyrrolocarbazole HOFFMANN LA ROCHE (CH) 1998-10-21 EP disclosed
US-5721267-A ANTICANCER AGENTS SYNTEX (U.S.A.) INC. (US) 1998-02-24 US disclosed
EP-0695755-A1 Pyrrolocarbazoles F. Hoffmann-La Roche AG (CH) 1996-02-07 EP disclosed