SCHEMBL8561865

SCHEMBL8561865

O=[N+]([O-])c1cccnc1C1CCNCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.44
PDE10A Q9Y233 1/20 0.44
CYP1A2 P05177 3/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 1/20 0.43
POLB P06746 1/20 0.43
ALDH1A1 P00352 5/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
PKM P14618 1/20 0.41
LMNA P02545 1/20 0.40
NCOA1 Q15788 1/20 0.40
NCOA3 Q9Y6Q9 1/20 0.40
HTR1A P08908 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
RAB9A P51151 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4439248 0.77 PDE10A (0.42) MAPTPDE10ACYP1A2CYP2C9CYP2C19
SCHEMBL8794324 0.76 MAPT (0.40) MAPTPDE10ACYP1A2CYP2C9CYP2C19
SCHEMBL8561395 0.76 HTR1A (0.49) HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL2093409 0.76 HTR1A (0.44) HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL8810623 0.75 CYP2C19 (0.46) MAPTPDE10ACYP1A2CYP2C9CYP2C19
SCHEMBL12124647 0.75 MAPT (0.45) MAPTPDE10ACYP1A2CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL15204558 0.74 MAPT (0.44) MAPTPDE10ACYP1A2CYP2C9CYP2C19
SCHEMBL20471758 0.74 ALDH1A1 (0.41) MAPTPDE10ACYP1A2CYP2C9CYP2C19
SCHEMBL28470144 0.74 MEN1 (0.51) MAPTPDE10ACYP1A2CYP2C9CYP2C19
SCHEMBL8748376 0.74 HTR2C (0.51) MAPTHTR1ASLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103415507-A 3-amino-pyridines as GPBAR1 agonists HOFFMANN LA ROCHE 2013-11-27 CN disclosed
EP-0735025-B1 Process for producing aminonitropyridines SUMITOMO CHEMICAL CO (JP) 1998-07-01 EP disclosed
US-5648496-A AMINATION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-07-15 US disclosed
CN-1138033-A Process for produducing aminonitropyridines SUMITOMO CHEMICAL CO (JP) 1996-12-18 CN disclosed
EP-0735025-A1 Process for producing aminonitropyridines SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1996-10-02 EP disclosed