SCHEMBL8748376

SCHEMBL8748376

O=[N+]([O-])c1ccccc1C1CCNCC1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 10/20 0.51
SLC6A2 P23975 5/20 0.45
SLC6A4 P31645 5/20 0.45
SLC6A3 Q01959 4/20 0.45
HTR1A P08908 3/20 0.45
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
SLC18A3 Q16572 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
ADRB2 P07550 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL227751 0.90 SLC6A2 (0.47) HTR2CSLC6A2SLC6A4KDM4EMEN1
SCHEMBL31525035 0.87 HSD17B10 (0.47) KDM4EMEN1GAAMAPTHTT
SCHEMBL3253975 0.87 HSD17B10 (0.47) KDM4EMEN1GAAMAPTHTT
SCHEMBL1065970 0.84 MEN1 (0.47) KDM4EMEN1GAAMAPTHTT
SCHEMBL28316412 0.84 ALDH1A1 (0.47) KDM4EMEN1GAAMAPTHTT
SCHEMBL7335158 0.82 HSP90AA1 (0.49) KDM4EMEN1GAAMAPTHTT
SCHEMBL3536567 0.81 HTR2C (0.50) HTR2CSLC6A2SLC6A4SLC6A3HTR1A
SCHEMBL2205192 0.81 HTR2C (0.50) HTR2CSLC6A2SLC6A4SLC6A3HTR1A
SCHEMBL8560822 0.78 MEN1 (0.43) HTR2CMEN1GAAMAPTHTT
Piperazine SCHEMBL27288925 0.77 HSD17B10 (0.52) HTR2CMEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1322196-A Naphthalenecarboxamides as tachykinin receptor antagonists ASTRA ZENECA N N (SE) 2001-11-14 CN disclosed
CN-1059668-C Process for preparing N-aliphatic substituted P-phenylenediamines MONSANTO CO (US) 2000-12-20 CN disclosed
EP-0641308-B1 PROCESS FOR PREPARING N-ALIPHATIC SUBSTITUTED P-PHENYLENEDIAMINES MONSANTO CO (US) 1997-03-12 EP disclosed
EP-0641308-A1 PROCESS FOR PREPARING N-ALIPHATIC SUBSTITUTED P-PHENYLENEDIAMINES. MONSANTO CO (US) 1995-03-08 EP disclosed
WO-1993024443-A1 PROCESS FOR PREPARING N-ALIPHATIC SUBSTITUTED P-PHENYLENEDIAMINES MONSANTO COMPANY (US) 1993-12-09 WO disclosed
US-5252737-A Process for preparing N-aliphatic substituted p-phenylenediamines MONSANTO COMPANY (US) 1993-10-12 US disclosed