SCHEMBL8561883

SCHEMBL8561883

Cc1ccc(-c2cc(Cl)ccc2C(N)=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.50
ALDH1A1 P00352 2/20 0.50
GLA P06280 1/20 0.50
GAA P10253 1/20 0.50
GRM2 Q14416 2/20 0.48
MAPT P10636 3/20 0.46
HPGD P15428 3/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
IKBKB O14920 3/20 0.44
CHUK O15111 3/20 0.44
BTK Q06187 2/20 0.44
DHODH Q02127 1/20 0.43
LMNA P02545 2/20 0.43
HTT P42858 2/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
PLA2G1B P04054 1/20 0.43
XBP1 P17861 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6492374 0.85 DHODH (0.55) KDM4EALDH1A1MAPTHPGDRAB9A
SCHEMBL17609420 0.83 BCAT2 (0.61) KDM4EALDH1A1GLAGAARAB9A
Hydrochloric Acid SCHEMBL5794611 0.82 P2RX1 (0.47) KDM4EALDH1A1GLAGAAIKBKB
SCHEMBL27259360 0.81 KLKB1 (0.52) KDM4EALDH1A1GLAGAAIKBKB
SCHEMBL5616388 0.80 GRM2 (0.48) GRM2IKBKBCHUKBTK
SCHEMBL28533539 0.77 DHODH (0.50) KDM4EALDH1A1GRM2MAPTHPGD
SCHEMBL5616523 0.77 CASP1 (0.46) KDM4EALDH1A1GLAGAARAB9A
SCHEMBL4067434 0.77 GRM2 (0.55) GRM2RAB9ANPC1IKBKBCHUK
SCHEMBL31541702 0.76 HDAC7 (0.66) RAB9ANPC1IKBKBCHUKPLA2G1B
SCHEMBL6490357 0.76 DHODH (0.60) KDM4EALDH1A1HPGDRAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0598702-B1 Biphenylmethane derivative, the use of it and pharmacological compositions containing same EISAI CO LTD (JP) 1998-06-10 EP disclosed
EP-0628557-B1 Biphenylmethane derivatives, the use of them and pharmacological compositions containing same EISAI CO LTD (JP) 1997-05-02 EP disclosed
US-5506238-A HYPOTENSIVE AGENT EISAI CO., LTD. (JP) 1996-04-09 US disclosed
EP-0420237-B1 Biphenylmethane derivative, the use of it and pharmacological compositions containing same EISAI CO LTD (JP) 1996-03-06 EP disclosed
EP-0628557-A1 Biphenylmethane derivatives, the use of them and pharmacological compositions containing same Eisai Co., Ltd. (JP) 1994-12-14 EP disclosed
US-5328911-A Cardiovascular disorders, hypotensive agents and congestive heart failure EISAI CO., LTD. (JP) 1994-07-12 US disclosed
EP-0598702-A1 Biphenylmethane derivative, the use of it and pharmacological compositions containing same Eisai Co., Ltd. (JP) 1994-05-25 EP disclosed
US-5298518-A Biphenylmethane derivative and pharmacological use EISAI CO., LTD. (JP) 1994-03-29 US disclosed
EP-0420237-A1 Biphenylmethane derivative, the use of it and pharmacological compositions containing same Eisai Co., Ltd. (JP) 1991-04-03 EP disclosed