SCHEMBL8562185

SCHEMBL8562185

CCOCCOCC[C@@](C)(O)Cc1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.37
MMP14 P50281 1/20 0.37
PTGS2 P35354 3/20 0.36
EPHX2 P34913 1/20 0.36
NR1H4 Q96RI1 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
CCR2 P41597 3/20 0.35
MMP1 P03956 1/20 0.34
MMP9 P14780 1/20 0.34
MMP13 P45452 1/20 0.34
ENPP2 Q13822 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8081741 0.78 ENPP2 (0.44) PTGS2EPHX2NR1H4PTGDR2ENPP2
SCHEMBL8077236 0.78 ENPP2 (0.44) PTGS2EPHX2NR1H4PTGDR2ENPP2
SCHEMBL8133933 0.72 ENPP2 (0.48) PTGS2EPHX2NR1H4ENPP2
SCHEMBL15836429 0.69 PTGS2 (0.53) MMP14PTGS2PTGDR2ENPP2
SCHEMBL2600037 0.69 ESR1 (0.50) PTGS2EPHX2NR1H4ENPP2
SCHEMBL8189822 0.68 MMP14 (0.36) GAAMMP14PTGS2ENPP2
SCHEMBL8189819 0.68 MMP14 (0.36) GAAMMP14PTGS2ENPP2
SCHEMBL29771215 0.68 CA12 (0.50) MMP14PTGS2MMP9MMP13
SCHEMBL18403162 0.68 EPHX2 (0.40) PTGS2EPHX2NR1H4ENPP2
SCHEMBL14462577 0.68 ENPP2 (0.42) PTGS2EPHX2NR1H4ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863891-A1 (METHYLSULFONYL)PHENYL-2-(5H)-FURANONES AS COX-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1998-09-16 EP disclosed
WO-1997014691-A1 (METHYLSULFONYL)PHENYL-2-(5H)-FURANONES AS COX-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1997-04-24 WO disclosed