SCHEMBL8562408

SCHEMBL8562408

O=C(O)CCc1ccc(N2CCN(c3ccc4c(c3)CCNCC4)C2=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.44
HTR6 P50406 8/20 0.43
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43
RXRG P48443 1/20 0.43
ITGB3 P05106 4/20 0.39
ITGA2B P08514 4/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
PRMT1 Q99873 1/20 0.38
ACHE P22303 1/20 0.38
ESR1 P03372 1/20 0.38
FFAR1 O14842 1/20 0.36
MLNR O43193 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8566413 0.94 RXRA (0.43) S1PR1HTR6RXRARXRBRXRG
SCHEMBL8557059 0.93 S1PR1 (0.43) S1PR1HTR6RXRARXRBRXRG
Hydrochloric Acid SCHEMBL8564109 0.92 S1PR1 (0.47) S1PR1HTR6RXRARXRBRXRG
Hydrochloric Acid SCHEMBL8559315 0.89 PRMT1 (0.43) HTR6PRMT1ACHE
Hydrochloric Acid SCHEMBL8564486 0.87 HTR6 (0.44) S1PR1HTR6RXRARXRBRXRG
SCHEMBL8559863 0.87 S1PR1 (0.50) S1PR1HTR6RXRARXRBRXRG
SCHEMBL8559578 0.87 HTR6 (0.42) S1PR1HTR6ACHEMLNR
SCHEMBL8560429 0.87 HTR6 (0.47) S1PR1HTR6RXRARXRBRXRG
Hydrochloric Acid SCHEMBL8559613 0.87 HTR6 (0.39) S1PR1HTR6RXRARXRBRXRG
Hydrochloric Acid SCHEMBL8563445 0.86 S1PR1 (0.49) S1PR1HTR6RXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP claimed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US claimed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP claimed
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed