SCHEMBL8560429

SCHEMBL8560429

O=C(O)CCc1ccc(N2CCN(c3ccc4c(c3)CCCNC4)C2=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.47
RXRA P19793 2/20 0.42
RXRB P28702 2/20 0.42
RXRG P48443 2/20 0.42
S1PR1 P21453 1/20 0.41
ITGB3 P05106 2/20 0.39
ITGA2B P08514 2/20 0.39
F10 P00742 3/20 0.38
ACHE P22303 1/20 0.38
ESR1 P03372 1/20 0.38
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
MCHR1 Q99705 1/20 0.36
CYP17A1 P05093 1/20 0.36
PRMT1 Q99873 1/20 0.36
FFAR1 O14842 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8557059 0.94 S1PR1 (0.43) HTR6RXRARXRBRXRGS1PR1
SCHEMBL8562408 0.87 S1PR1 (0.44) HTR6RXRARXRBRXRGS1PR1
Hydrochloric Acid SCHEMBL8566413 0.84 RXRA (0.43) HTR6RXRARXRBRXRGS1PR1
SCHEMBL8563370 0.81 ASIC3 (0.40) HTR6S1PR1F10
SCHEMBL8559863 0.81 S1PR1 (0.50) HTR6RXRARXRBRXRGS1PR1
Acetic Acid SCHEMBL8895876 0.81 ASIC3 (0.38) HTR6S1PR1ITGB3ITGA2BF10
Hydrochloric Acid SCHEMBL8563445 0.80 S1PR1 (0.49) HTR6RXRARXRBRXRGS1PR1
Hydrochloric Acid SCHEMBL8564109 0.80 S1PR1 (0.47) HTR6RXRARXRBRXRGS1PR1
SCHEMBL8559326 0.78 S1PR1 (0.47) RXRARXRBRXRGS1PR1ITGB3
SCHEMBL8560495 0.78 HTR6 (0.43) HTR6RXRARXRBRXRGITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed