SCHEMBL8562449

SCHEMBL8562449

O=C(Nc1ccc(C(=O)N2c3ccccc3CNc3ccccc32)cc1)c1ccccc1C(F)(F)F

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 3/20 0.46
AVPR1A P37288 3/20 0.46
KCNK3 O14649 1/20 0.43
KCNK9 Q9NPC2 1/20 0.43
AURKA O14965 1/20 0.43
AURKB Q96GD4 1/20 0.43
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
PTPRC P08575 1/20 0.41
PTGS1 P23219 1/20 0.41
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
OXTR P30559 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559885 0.93 AVPR2 (0.46) AVPR2AVPR1AKCNK3KCNK9AURKA
SCHEMBL8559861 0.90 AURKA (0.47) AVPR2AVPR1AAURKAAURKB
SCHEMBL8557883 0.87 MEN1 (0.50) AVPR2AVPR1ALMNATP53
SCHEMBL8562616 0.87 ITGB1 (0.40) AVPR2AVPR1ATP53
SCHEMBL8558194 0.86 AKT1 (0.52) AURKALMNATP53
SCHEMBL8556562 0.86 KCNK3 (0.44) AVPR2AVPR1AKCNK3KCNK9RXFP1
SCHEMBL8559901 0.85 AVPR2 (0.63) AVPR2AVPR1AOXTR
SCHEMBL8560617 0.85 AVPR1A (0.49) AVPR2AVPR1ALMNA
SCHEMBL8557851 0.84 MAPT (0.48) AVPR2AVPR1AAURKALMNATP53
SCHEMBL8557390 0.83 AVPR2 (0.52) AVPR2AVPR1AOXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed