SCHEMBL8562616

SCHEMBL8562616

O=C(Nc1ccc(C(=O)N2c3ccccc3CNc3ccccc32)cc1)c1c(F)cccc1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 2/20 0.40
ITGA4 P13612 2/20 0.40
AKT1 P31749 1/20 0.39
TYK2 P29597 2/20 0.38
AVPR2 P30518 1/20 0.37
AVPR1A P37288 1/20 0.37
RORC P51449 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
HTT P42858 1/20 0.36
NOD2 Q9HC29 1/20 0.36
TP53 P04637 1/20 0.36
CNR1 P21554 2/20 0.36
CNR2 P34972 2/20 0.36
ACKR3 P25106 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562699 0.88 AVPR2 (0.39) ITGB1ITGA4AKT1AVPR2AVPR1A
SCHEMBL8559885 0.87 AVPR2 (0.46) AVPR2AVPR1A
SCHEMBL8562449 0.87 AVPR2 (0.46) AVPR2AVPR1ATP53
SCHEMBL8558246 0.86 AVPR2 (0.48) ITGB1ITGA4TYK2AVPR2AVPR1A
SCHEMBL8558194 0.86 AKT1 (0.52) AKT1TP53
SCHEMBL8559231 0.84 AVPR2 (0.49) TYK2AVPR2AVPR1AKMT2AJAK2
SCHEMBL8557883 0.84 MEN1 (0.50) AKT1AVPR2AVPR1AMEN1KMT2A
SCHEMBL8559861 0.83 AURKA (0.47) AKT1AVPR2AVPR1A
SCHEMBL8556942 0.82 NPC1 (0.49) MEN1KMT2AHTTTP53
SCHEMBL8562066 0.82 AURKA (0.47) AKT1AVPR2AVPR1AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed