SCHEMBL8562680

SCHEMBL8562680

O=C(Nc1ccc(C(=O)N2CCc3ccccc3-c3ccccc32)cc1)c1ccccc1

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.59
HPGD P15428 1/20 0.59
AVPR2 P30518 2/20 0.58
AVPR1A P37288 2/20 0.58
OXTR P30559 1/20 0.58
RAB9A P51151 1/20 0.58
NAMPT P43490 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556989 0.85 AVPR1A (0.72) AVPR2AVPR1AOXTR
SCHEMBL8559975 0.85 AVPR2 (0.58) HPGDAVPR2AVPR1AOXTRRAB9A
SCHEMBL8556457 0.85 AVPR2 (0.58) AVPR2AVPR1AOXTRNAMPT
SCHEMBL8562670 0.85 AVPR1A (0.60) AVPR2AVPR1AOXTR
SCHEMBL8560388 0.85 AVPR1A (0.60) AVPR2AVPR1AOXTRNAMPT
SCHEMBL8561545 0.85 MEN1 (0.74) AVPR2AVPR1AOXTRRAB9ANAMPT
SCHEMBL8558667 0.84 NAMPT (0.54) ALDH1A1HPGDAVPR2AVPR1AOXTR
SCHEMBL8557460 0.84 AVPR1A (0.64) AVPR2AVPR1AOXTR
SCHEMBL7345982 0.83 RAB9A (0.78) RAB9A
SCHEMBL8557218 0.83 AVPR1A (0.60) ALDH1A1AVPR2AVPR1AOXTRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed