SCHEMBL8562916

SCHEMBL8562916

CN1CCc2ccc(N3CC(=O)N(C4CCC(CCC(=O)O)CC4)C3=O)cc2CC1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.38
DRD3 P35462 5/20 0.38
PTGER3 P43115 1/20 0.37
PTGER2 P43116 1/20 0.37
DRD2 P14416 9/20 0.35
HRH1 P35367 3/20 0.35
HTR2A P28223 1/20 0.35
ACHE P22303 2/20 0.35
TMEM97 Q5BJF2 2/20 0.33
SIGMAR1 Q99720 2/20 0.33
DGAT1 O75907 1/20 0.33
F10 P00742 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRK1 P41145 1/20 0.33
OPRL1 P41146 1/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561989 1.00 HTR1A (0.38) HTR1ADRD3PTGER3PTGER2DRD2
Hydrochloric Acid SCHEMBL8985722 0.99 HTR1A (0.37) HTR1ADRD3PTGER3PTGER2DRD2
Hydrochloric Acid SCHEMBL8560651 0.99 HTR1A (0.37) HTR1ADRD3PTGER3PTGER2DRD2
Hydrochloric Acid SCHEMBL8564536 0.87 HTR6 (0.42) PTGER3PTGER2ACHE
SCHEMBL8562349 0.85 F2 (0.39) ACHEDGAT1F10
SCHEMBL8562341 0.85 F2 (0.39) ACHEDGAT1F10
Hydrochloric Acid SCHEMBL8560749 0.84 F2 (0.38) ACHEDGAT1F10
Hydrochloric Acid SCHEMBL8566388 0.83 F10 (0.36) DRD2ACHETMEM97SIGMAR1DGAT1
SCHEMBL8562636 0.83 F10 (0.40) ACHEF10
SCHEMBL8562641 0.83 F10 (0.40) ACHEF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP claimed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP claimed
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed