SCHEMBL8562929

SCHEMBL8562929

CC(=O)Nc1cc(Cl)ncc1NS(=O)(=O)C(C)=O

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
CA9 Q16790 3/20 0.38
PTK2 Q05397 1/20 0.36
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
PIK3CD O00329 1/20 0.36
PIK3CG P48736 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
KDM4E B2RXH2 2/20 0.35
HSD17B10 Q99714 1/20 0.35
ALDH1A1 P00352 3/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
PIK3C3 Q8NEB9 2/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
PGK1 P00558 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561506 0.81 PIK3CD (0.35) CA1CA2CA9KMT2AMEN1
SCHEMBL21672318 0.76 PGK1 (0.45) CA1CA2CA9PTK2KMT2A
SCHEMBL30456319 0.76 ALDH1A1 (0.46) CA1CA2CA9PTK2KMT2A
SCHEMBL18130725 0.74 NPC1 (0.47) PTK2KDM4EHSD17B10ALDH1A1L3MBTL1
SCHEMBL25604920 0.74 ALDH1A1 (0.43) PTK2KMT2AMEN1KDM4EHSD17B10
SCHEMBL9261109 0.73 KMT2A (0.41) CA1CA2CA9PTK2KMT2A
Acetic Acid SCHEMBL28092089 0.73 ALDH1A1 (0.44) CA1CA2CA9PTK2KMT2A
SCHEMBL16441504 0.73 PTK2 (0.41) CA1CA2CA9PTK2KMT2A
SCHEMBL17059904 0.68 MEN1 (0.44) CA1CA2CA9KMT2AMEN1
SCHEMBL11816879 0.65 TRPV1 (0.50) KMT2AMEN1KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618209-B1 Pyridothiadiazines, processes for their preparation and pharmaceutical compositions containing them ADIR (FR) 1998-12-23 EP disclosed
EP-0618209-A1 Pyridothiadiazines, processes for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1994-10-05 EP disclosed