SCHEMBL8562987

SCHEMBL8562987

COc1ccc(CNC(=O)[C@@H](Br)CCBr)cc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
HPGD P15428 3/20 0.50
PKM P14618 1/20 0.50
GAA P10253 1/20 0.49
CASR P41180 1/20 0.49
NPC1 O15118 4/20 0.49
RAB9A P51151 3/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
ANPEP P15144 1/20 0.48
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562984 1.00 ALDH1A1 (0.51) ALDH1A1KMT2AMEN1HPGDPKM
SCHEMBL27554758 0.85 ALDH1A1 (0.64) ALDH1A1KMT2AMEN1HPGDPKM
SCHEMBL8561177 0.84 ALDH1A1 (0.56) ALDH1A1KMT2AMEN1HPGDGAA
SCHEMBL8561171 0.84 ALDH1A1 (0.56) ALDH1A1KMT2AMEN1HPGDGAA
SCHEMBL16885994 0.84 KMT2A (0.54) ALDH1A1KMT2AMEN1HPGDPKM
SCHEMBL11735404 0.82 ALDH1A1 (0.59) ALDH1A1KMT2AMEN1HPGDPKM
SCHEMBL1543096 0.81 MEN1 (0.54) ALDH1A1KMT2AMEN1HPGDGAA
SCHEMBL8562678 0.81 HPGD (0.49) ALDH1A1KMT2AHPGDGAANPC1
SCHEMBL8562675 0.81 HPGD (0.49) ALDH1A1KMT2AHPGDGAANPC1
SCHEMBL8568656 0.80 MMP8 (0.51) ALDH1A1KMT2AMEN1PKMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5804577-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1998-09-08 US disclosed
EP-0761673-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed