SCHEMBL8563028

SCHEMBL8563028

COC(=O)CCC1(c2ccccc2)CNC(=O)N1c1ccc2c(c1)CCNCC2

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 8/20 0.37
NOTUM Q6P988 1/20 0.33
ACHE P22303 1/20 0.33
MCHR1 Q99705 1/20 0.33
DRD2 P14416 2/20 0.33
DRD1 P21728 2/20 0.33
DRD4 P21917 1/20 0.33
DRD5 P21918 1/20 0.33
DRD3 P35462 1/20 0.33
HTR2C P28335 3/20 0.32
HTR2B P41595 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8559380 0.99 HTR6 (0.36) HTR6NOTUMACHEMCHR1DRD2
SCHEMBL8563449 0.94 HTR6 (0.36) HTR6NOTUM
SCHEMBL8559515 0.91 HTR6 (0.39) HTR6NOTUMDRD2DRD1DRD4
SCHEMBL8558612 0.90 NOTUM (0.36) HTR6NOTUMACHEMCHR1DRD2
Hydrochloric Acid SCHEMBL8563487 0.90 HTR6 (0.39) HTR6NOTUMDRD2DRD1DRD4
Hydrochloric Acid SCHEMBL8565214 0.89 NOTUM (0.36) HTR6NOTUMACHEMCHR1DRD2
Hydrochloric Acid SCHEMBL8559768 0.85 ALDH1A1 (0.36) HTR6ACHEMCHR1DRD2DRD1
SCHEMBL8566144 0.84 PTGER1 (0.34) HTR6
Hydrochloric Acid SCHEMBL8557445 0.83 PTGER1 (0.35) HTR6
SCHEMBL8560509 0.81 TMEM97 (0.42) HTR6NOTUMHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed