SCHEMBL8563249

SCHEMBL8563249

CN(C(=O)c1cc(Cl)ccc1Cl)c1ccc(C(=O)N2Cc3ccccc3Cc3ccccc32)cc1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 5/20 0.48
AVPR1A P37288 4/20 0.48
HSD17B3 P37058 2/20 0.42
LMNA P02545 1/20 0.41
HSP90AA1 P07900 1/20 0.40
PDK1 Q15118 1/20 0.40
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562797 0.92 AVPR2 (0.54) AVPR2AVPR1AHSD17B3HSP90AA1PDK1
SCHEMBL8561048 0.90 AVPR2 (0.48) AVPR2AVPR1AHSD17B3HSP90AA1PDK1
SCHEMBL8559548 0.90 POLB (0.51) AVPR2AVPR1ALMNAHSP90AA1PDK1
SCHEMBL8559862 0.87 AVPR2 (0.45) AVPR2AVPR1AHSD17B3HSP90AA1PDK1
SCHEMBL8557534 0.85 AVPR2 (0.45) AVPR2AVPR1AHSP90AA1PDK1POLB
SCHEMBL7336560 0.84 AVPR1A (0.62) AVPR2AVPR1A
SCHEMBL8561629 0.83 AVPR2 (0.52) AVPR2AVPR1A
SCHEMBL8558249 0.82 NPC1 (0.45) AVPR2AVPR1AHSP90AA1PDK1
SCHEMBL8561685 0.82 AVPR1A (0.44) AVPR2AVPR1AHSP90AA1PDK1
SCHEMBL8558027 0.80 AVPR2 (0.69) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed