SCHEMBL8559862

SCHEMBL8559862

COc1cc(Cl)ccc1C(=O)N(C)c1ccc(C(=O)N2Cc3ccccc3Cc3ccccc32)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 5/20 0.45
AVPR1A P37288 5/20 0.45
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40
TUBA4A P68366 1/20 0.40
TUBB4B P68371 1/20 0.40
TUBB3 Q13509 1/20 0.40
TUBB2A Q13885 1/20 0.40
TUBB8 Q3ZCM7 1/20 0.40
TUBA3E Q6PEY2 1/20 0.40
TUBA1A Q71U36 1/20 0.40
TUBA1C Q9BQE3 1/20 0.40
TUBB6 Q9BUF5 1/20 0.40
TUBB2B Q9BVA1 1/20 0.40
TUBB1 Q9H4B7 1/20 0.40
HSP90AA1 P07900 1/20 0.40
PDK1 Q15118 1/20 0.40
PDE4A P27815 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561776 0.90 SMN1; SMN2 (0.46) AVPR2AVPR1ATUBB4ATUBBTUBA3C
SCHEMBL8561048 0.89 AVPR2 (0.48) AVPR2AVPR1AHSP90AA1PDK1HSD17B3
SCHEMBL8562797 0.89 AVPR2 (0.54) AVPR2AVPR1AHSP90AA1PDK1HSD17B3
SCHEMBL8557707 0.89 ALDH1A1 (0.47) AVPR2AVPR1ATUBB4ATUBBTUBA3C
SCHEMBL8563249 0.87 AVPR2 (0.48) AVPR2AVPR1AHSP90AA1PDK1HSD17B3
SCHEMBL7341415 0.85 AVPR1A (0.63) AVPR2AVPR1A
SCHEMBL8559548 0.83 POLB (0.51) AVPR2AVPR1AHSP90AA1PDK1ALDH1A1
SCHEMBL8557743 0.83 AVPR2 (0.64) AVPR2AVPR1AACHE
SCHEMBL8557534 0.82 AVPR2 (0.45) AVPR2AVPR1AHSP90AA1PDK1RAB9A
SCHEMBL8558249 0.81 NPC1 (0.45) AVPR2AVPR1AHSP90AA1PDK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed