SCHEMBL8563530

SCHEMBL8563530

CCOc1cc2c(Cl)c(Br)cnc2nc1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
ENPP1 P22413 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
S1PR1 P21453 3/20 0.34
CYP1A2 P05177 2/20 0.33
CYP2C19 P33261 2/20 0.33
KDM4E B2RXH2 2/20 0.33
LMNA P02545 1/20 0.33
GRM5 P41594 2/20 0.32
TSHR P16473 2/20 0.32
HSD17B10 Q99714 1/20 0.32
AOC3 Q16853 2/20 0.32
S1PR3 Q99500 2/20 0.32
MAPT P10636 2/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
HPGD P15428 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563128 0.85 KDM4E (0.37) ALDH1A1ENPP1S1PR1CYP1A2CYP2C19
SCHEMBL8561182 0.84 HSD17B10 (0.36) ALDH1A1ADORA2AADORA1S1PR1CYP1A2
SCHEMBL8326771 0.80 SRC (0.42) KDM4EMAPTTDP1L3MBTL1GAA
SCHEMBL8326372 0.79 TSHR (0.40) ALDH1A1CYP1A2KDM4ELMNATSHR
SCHEMBL8327645 0.78 KMT2A (0.51) ALDH1A1KDM4ETSHRMAPTHPGD
SCHEMBL8326185 0.78 SLC2A1 (0.40) LMNATSHRDPP4
SCHEMBL8565727 0.75 KDM4E (0.33) ALDH1A1ADORA1CYP1A2CYP2C19KDM4E
SCHEMBL8321420 0.74 SMN1; SMN2 (0.39) ALDH1A1ENPP1CYP1A2CYP2C19KDM4E
SCHEMBL8566080 0.72 PDE4B (0.43) KDM4EMAPTL3MBTL1GAA
SCHEMBL8567944 0.72 KDM4E (0.38) ALDH1A1ENPP1ADORA2AADORA1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618916-B1 ANTI-RHEUMATIC NAPHTHYRIDINE DERIVATIVES KNOLL AG (DE) 1998-09-23 EP disclosed
US-5464781-A TREATING RHEUMATIC DISEASES THE BOOTS COMPANY PLC (GB) 1995-11-07 US disclosed