SCHEMBL8563585

SCHEMBL8563585

CCCn1c2nc(-c3ccco3)[nH]c2c(=O)n2nc(-c3ccco3)nc12

nearest known ligand 0.71

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 6/20 0.54
ADORA2A P29274 4/20 0.54
ADORA3 P0DMS8 1/20 0.50
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
KMT2A Q03164 1/20 0.48
HSD17B10 Q99714 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8872400 0.84 ADORA2B (0.69) ADORA2BADORA2AKDM4EMEN1ALDH1A1
SCHEMBL6995974 0.82 MEN1 (0.49) ADORA2BADORA2AADORA3MEN1CYP1A2
SCHEMBL6997253 0.80 ADORA2A (0.48) ADORA2BADORA2AADORA3
SCHEMBL5230763 0.74 ADORA2B (0.52) ADORA2BADORA2AADORA3KDM4EMEN1
SCHEMBL10673069 0.71 KDM4E (0.64) ADORA2BADORA2AADORA3KDM4EALDH1A1
SCHEMBL2686441 0.71 ADORA2B (0.52) ADORA2BADORA2AADORA3KDM4EMEN1
SCHEMBL1720432 0.71 ADORA2A (0.51) ADORA2BADORA2AADORA3KDM4EMEN1
SCHEMBL5620839 0.67 ADORA2B (0.54) ADORA2BADORA2AKDM4EMEN1ALDH1A1
SCHEMBL25539381 0.66 ADORA2A (0.58) ADORA2BADORA2AADORA3
SCHEMBL661108 0.66 ADORA2B (1.00) ADORA2BADORA2AADORA3KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880524-A1 NEW TRIAZOLOPURINES, METHOD OF PREPARING THEM AND THEIR USE AS DRUGS Boehringer Ingelheim Pharma KG (DE) 1998-12-02 EP disclosed
WO-1998003511-A1 NEW TRIAZOLOPURINES, METHOD OF PREPARING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-01-29 WO disclosed