SCHEMBL8563778

SCHEMBL8563778

CNS(=O)(=O)c1ccc(O)c(C(C)=O)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.50
KDM4E B2RXH2 4/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
POLB P06746 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.46
SERPINE1 P05121 1/20 0.46
ALDH1A1 P00352 4/20 0.45
HSD17B10 Q99714 3/20 0.45
HPGD P15428 2/20 0.45
GAA P10253 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA3 P07451 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43
CA5A P35218 1/20 0.43
CA7 P43166 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2825786 0.86 ALDH1A1 (0.62) LMNAKDM4EMEN1KMT2APOLB
SCHEMBL1520426 0.85 KDM4E (0.58) LMNAKDM4EMEN1KMT2APOLB
SCHEMBL2828647 0.83 MEN1 (0.58) LMNAKDM4EMEN1KMT2APOLB
SCHEMBL11183233 0.81 VCAM1 (0.54) LMNAMEN1KMT2AL3MBTL1ALDH1A1
SCHEMBL1577295 0.80 LMNA (0.51) LMNAKDM4EMEN1KMT2APOLB
SCHEMBL7143573 0.80 CA1 (0.55) KDM4EMEN1KMT2AALDH1A1HSD17B10
SCHEMBL312086 0.80 HSD17B10 (0.68) LMNAKDM4EMEN1KMT2APOLB
SCHEMBL9143971 0.80 SERPINE1 (0.70) LMNAL3MBTL1SERPINE1ALDH1A1GAA
Ammonia Solution, Strong SCHEMBL7644798 0.79 HSD17B10 (0.66) LMNAKDM4EMEN1KMT2APOLB
Ammonia Solution, Strong SCHEMBL7644790 0.79 HSD17B10 (0.66) LMNAKDM4EMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP disclosed
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
CN-1110685-A Nitrogen-containing spiro ring MERCK & CO INC (US) 1995-10-25 CN disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
CN-1053613-A Nitrogen-containing spiro ring MERCK & CO INC (US) 1991-08-07 CN disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed