SCHEMBL8564137

SCHEMBL8564137

Nc1nc(N)c2c(ccn2CCCc2ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s2)n1

nearest known ligand 0.75

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ATIC P31939 12/20 0.75
SHMT1 P34896 10/20 0.75
SHMT2 P34897 10/20 0.75
GART P22102 13/20 0.71
FOLR1 P15328 9/20 0.53
FOLR2 P14207 3/20 0.51
SLC46A1 Q96NT5 6/20 0.51
SLC19A1 P41440 4/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8564142 1.00 ATIC (0.75) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL8569348 0.95 ATIC (0.67) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL8569343 0.95 ATIC (0.67) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL9001788 0.86 ATIC (1.00) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL20854930 0.86 ATIC (1.00) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL8565091 0.85 ATIC (0.55) ATICSHMT1SHMT2GART
SCHEMBL8565081 0.85 ATIC (0.55) ATICSHMT1SHMT2GART
SCHEMBL8563875 0.84 ATIC (0.74) ATICSHMT1SHMT2GART
SCHEMBL8563883 0.84 ATIC (0.74) ATICSHMT1SHMT2GART
SCHEMBL8570075 0.84 ATIC (0.54) ATICSHMT1SHMT2GART

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed