SCHEMBL8569348

SCHEMBL8569348

Nc1nc(N)c2c(ccn2CCc2ccc(C(=O)N[C@H](CCC(=O)O)C(=O)O)s2)n1

nearest known ligand 0.67

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ATIC P31939 11/20 0.67
SHMT1 P34896 9/20 0.67
SHMT2 P34897 9/20 0.67
GART P22102 13/20 0.66
FOLR1 P15328 10/20 0.51
SLC46A1 Q96NT5 7/20 0.49
SLC19A1 P41440 5/20 0.49
FOLR2 P14207 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8569343 1.00 ATIC (0.67) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL8564137 0.95 ATIC (0.75) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL8564142 0.95 ATIC (0.75) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL8565081 0.87 ATIC (0.55) ATICSHMT1SHMT2GART
SCHEMBL8565091 0.87 ATIC (0.55) ATICSHMT1SHMT2GART
SCHEMBL8570075 0.85 ATIC (0.54) ATICSHMT1SHMT2GART
SCHEMBL9001824 0.85 ATIC (0.91) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL8570081 0.85 ATIC (0.54) ATICSHMT1SHMT2GART
SCHEMBL8570220 0.84 ATIC (0.52) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL8570214 0.84 ATIC (0.52) ATICSHMT1SHMT2GARTFOLR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed