SCHEMBL8565091

SCHEMBL8565091

C=C(CCn1ccc2nc(N)nc(N)c21)c1ccc(C(=O)N[C@H](CCC(=O)O)C(=O)O)s1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ATIC P31939 14/20 0.55
SHMT1 P34896 14/20 0.55
SHMT2 P34897 14/20 0.55
GART P22102 11/20 0.55
DHFR P00374 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8565081 1.00 ATIC (0.55) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8570214 0.92 ATIC (0.52) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8570220 0.92 ATIC (0.52) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8563429 0.88 ATIC (0.56) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8563442 0.88 ATIC (0.56) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8569343 0.87 ATIC (0.67) ATICSHMT1SHMT2GART
SCHEMBL8569348 0.87 ATIC (0.67) ATICSHMT1SHMT2GART
SCHEMBL9001783 0.85 ATIC (0.75) ATICSHMT1SHMT2GART
SCHEMBL8564142 0.85 ATIC (0.75) ATICSHMT1SHMT2GART
SCHEMBL8564137 0.85 ATIC (0.75) ATICSHMT1SHMT2GART

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed