SCHEMBL8564297

SCHEMBL8564297

CC(C)(C)NC(=O)c1ccc(N2CCN(c3ccncc3)CC2I)cc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.38
POLB P06746 1/20 0.38
HPGD P15428 1/20 0.38
MAPT P10636 2/20 0.38
DRD2 P14416 1/20 0.36
AURKA O14965 1/20 0.36
TTK P33981 1/20 0.36
AURKB Q96GD4 1/20 0.36
INCENP Q9NQS7 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
USP2 O75604 1/20 0.35
TP53 P04637 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7956169 0.84 SLC2A1 (0.51) SLC2A1SMN1; SMN2POLBHPGDMAPT
SCHEMBL8565666 0.74 MAPT (0.40) SMN1; SMN2POLBMAPTALDH1A1GAA
SCHEMBL15448546 0.71 HDAC3 (0.61) SMN1; SMN2TP53
SCHEMBL1423877 0.70 SMN1; SMN2 (0.67) SMN1; SMN2POLBHPGDALDH1A1GAA
SCHEMBL25753493 0.70 HDAC6 (0.63) SMN1; SMN2HPGDMAPTALDH1A1GAA
SCHEMBL7961490 0.70 MAPT (0.54) SLC2A1SMN1; SMN2MAPTDRD2AURKA
SCHEMBL13701825 0.69 MAPT (0.64) SMN1; SMN2POLBHPGDMAPTALDH1A1
SCHEMBL8635363 0.65 SLC2A1 (0.45) SLC2A1SMN1; SMN2MAPTGAATP53
SCHEMBL17865779 0.65 LMNA (0.58) SMN1; SMN2POLBMAPT
SCHEMBL7956272 0.65 NPC1 (0.69) SMN1; SMN2MAPTALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880501-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1998-12-02 EP disclosed
WO-1997028128-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1997-08-07 WO disclosed