SCHEMBL8564350

SCHEMBL8564350

Cc1cc(OCOc2ccc(N=C=O)c(C)c2)ccc1N=C=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.43
TRPA1 O75762 1/20 0.43
TDP1 Q9NUW8 3/20 0.41
HPGD P15428 3/20 0.41
ALDH1A1 P00352 2/20 0.41
PDIA6 Q15084 1/20 0.35
MCL1 Q07820 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.33
ESR1 P03372 1/20 0.33
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33
APEX1 P27695 1/20 0.33
MAPK1 P28482 1/20 0.33
ESR2 Q92731 1/20 0.33
MAPT P10636 2/20 0.32
ATM Q13315 1/20 0.32
RAB9A P51151 2/20 0.31
MEN1 O00255 1/20 0.31
PKM P14618 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8567728 0.92 CYP3A4 (0.49) CYP3A4TRPA1TDP1HPGDALDH1A1
SCHEMBL10341831 0.90 CYP3A4 (0.43) CYP3A4TRPA1TDP1HPGDALDH1A1
SCHEMBL10697590 0.88 CYP3A4 (0.42) CYP3A4TRPA1TDP1HPGDALDH1A1
SCHEMBL10341987 0.88 PDIA6 (0.47) CYP3A4TRPA1TDP1HPGDALDH1A1
SCHEMBL8565996 0.87 CYP3A4 (0.36) CYP3A4TRPA1TDP1HPGDALDH1A1
SCHEMBL9918950 0.83 ALDH1A1 (0.46) CYP3A4TRPA1TDP1HPGDALDH1A1
SCHEMBL10341851 0.83 CYP3A4 (0.49) CYP3A4TRPA1TDP1HPGDALDH1A1
SCHEMBL162798 0.82 CYP3A4 (0.51) CYP3A4TRPA1TDP1HPGDALDH1A1
SCHEMBL10341870 0.82 CYP3A4 (0.47) CYP3A4TRPA1TDP1HPGDALDH1A1
SCHEMBL10038435 0.78 CYP3A4 (0.42) CYP3A4TRPA1TDP1HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731399-A OXYALKYLATION TO PRODUCT HYDROXY COMPOUND; PHOSGENATION TO PRODUCT POLYISOCYANATE COMPOUND IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1998-03-24 US disclosed
EP-0611050-B1 Polyol compositions and polyisocyanates for use in the preparation of polyurethanes ICI PLC (GB) 1997-06-18 EP disclosed
EP-0611050-A1 Novel di- and polyamino compounds for use in the preparation of polyurethanes IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-08-17 EP disclosed