SCHEMBL8565583

SCHEMBL8565583

CCOC(=O)[CH]CC(C)N(C)C

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 10/20 0.43
CHRNA4 P43681 10/20 0.43
CHRNB4 P30926 8/20 0.43
CHRNA3 P32297 7/20 0.43
HCAR2 Q8TDS4 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
ALDH1A1 P00352 2/20 0.34
MAPT P10636 1/20 0.33
LMNA P02545 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL128591 0.79 HCAR2 (0.45) HCAR2NPSR1ALDH1A1MAPTLMNA
SCHEMBL20028538 0.69 MGAM (0.46) CHRNB2CHRNA4CHRNB4CHRNA3ALDH1A1
SCHEMBL128754 0.69
SCHEMBL25585756 0.69 HCAR2 (0.48) CHRNB2CHRNA4CHRNB4CHRNA3HCAR2
SCHEMBL30929696 0.69 HCAR2 (0.48) CHRNB2CHRNA4CHRNB4CHRNA3HCAR2
SCHEMBL25537052 0.69 HCAR2 (0.48) CHRNB2CHRNA4CHRNB4CHRNA3HCAR2
SCHEMBL25537058 0.69 HCAR2 (0.48) CHRNB2CHRNA4CHRNB4CHRNA3HCAR2
SCHEMBL127141 0.68 HCAR2 (0.42) HCAR2NPSR1ALDH1A1MAPTLMNA
SCHEMBL1260437 0.68
SCHEMBL196972 0.66 ALDH1A1 (0.43) CHRNB2CHRNA4CHRNB4CHRNA3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0823908-A1 PYRIDO 2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1998-02-18 EP disclosed
WO-1996034867-A1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1996-11-07 WO disclosed