SCHEMBL8565717

SCHEMBL8565717

COC(=O)C(CN(C)Cc1ccc(Cl)c(Cl)c1)NC(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.42
KLK5 Q9Y337 1/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
KMT2A Q03164 1/20 0.41
PPARA Q07869 3/20 0.40
PPARG P37231 2/20 0.40
PSEN1 P49768 2/20 0.40
PSEN2 P49810 2/20 0.40
APH1B Q8WW43 2/20 0.40
NCSTN Q92542 2/20 0.40
APH1A Q96BI3 2/20 0.40
PSENEN Q9NZ42 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
CACNA1B Q00975 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560370 0.90 PPARA (0.47) TSHRMEN1LMNAKMT2APPARA
SCHEMBL30703902 0.83 PSEN1 (0.54) KLK5PPARAPPARGPSEN1PSEN2
SCHEMBL8560272 0.81 PSEN1 (0.46) KLK5PPARAPPARGPSEN1PSEN2
SCHEMBL8559055 0.80 TSHR (0.50) TSHRKLK5LMNAPPARAPPARG
SCHEMBL29839160 0.77 CTSL (0.48) TSHRPPARAPPARGCTSLTACR1
SCHEMBL27228870 0.77 CTSL (0.48) TSHRPPARAPPARGCTSLTACR1
SCHEMBL27228877 0.77 CTSL (0.48) TSHRPPARAPPARGCTSLTACR1
SCHEMBL27232298 0.77 CTSL (0.48) TSHRPPARAPPARGCTSLTACR1
SCHEMBL18130491 0.76 MEN1 (0.48) TSHRMEN1LMNAKMT2APPARA
SCHEMBL1311165 0.76 ACE (0.59) PPARAPPARGCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811431-A Spiro-substituted azacyclic derivatives and their use as therapeutic agents MERCK SHARP & DOHME LTD. (GB) 1998-09-22 US disclosed