SCHEMBL8560272

SCHEMBL8560272

COC(=O)C(CN(Cc1ccc(Cl)c(Cl)c1)C(=O)OCc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 6/20 0.46
PSEN2 P49810 6/20 0.46
APH1B Q8WW43 6/20 0.46
NCSTN Q92542 6/20 0.46
APH1A Q96BI3 6/20 0.46
PSENEN Q9NZ42 6/20 0.46
PPARA Q07869 3/20 0.46
KLK5 Q9Y337 1/20 0.44
BACE1 P56817 4/20 0.44
PPARG P37231 2/20 0.42
CTSS P25774 1/20 0.41
KYNU Q16719 1/20 0.41
SYK P43405 1/20 0.41
NOS2 P35228 1/20 0.41
ACE P12821 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562043 0.94 PPARA (0.51) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8565717 0.81 TSHR (0.42) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6089700 0.80 PPARA (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7822488 0.79 CTSL (0.44) PPARAKLK5CTSSACE
SCHEMBL8893110 0.77 PPARA (0.54) PPARAPPARGCTSSSYKACE
SCHEMBL8893121 0.77 PPARA (0.54) PPARAPPARGCTSSSYKACE
SCHEMBL20364471 0.75 KYNU (0.49) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8560370 0.74 PPARA (0.47) PPARAPPARGCTSSACE
SCHEMBL15122799 0.74 KYNU (0.48) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL15122801 0.74 KYNU (0.48) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811431-A Spiro-substituted azacyclic derivatives and their use as therapeutic agents MERCK SHARP & DOHME LTD. (GB) 1998-09-22 US disclosed